Submission Details
Molecule(s):
O=C1CCCN1Cc1cccc(C(=O)N2CCC(C3CCNC3)CC2)c1
Cc1ccc(Nc2ccccc2C(=O)N2CCC(C3CCNC3)CC2)cc1
CS(=O)(=O)Nc1ccc(Cl)cc1C(=O)N1CCC(C2CCNC2)CC1
O=C1CCc2cc(C(=O)N3CCC(C4CCNC4)CC3)ccc2N1
Cc1cc(C(=O)N2CCC(C3CCNC3)CC2)cc(S(=O)(=O)N(C)C)c1C
Cc1c(C(=O)N2CCC(C3CCNC3)CC2)cccc1-c1ccccn1
CCCOc1c(Cl)cc(C(=O)N2CCC(C3CCNC3)CC2)cc1OCC
CC(C)OCc1cc(C(=O)N2CCC(C3CCNC3)CC2)ccc1F
O=C(c1cccc(N2CCCNC2=O)c1)N1CCC(C2CCNC2)CC1
CN1CCN(c2ccc(F)cc2C(=O)N2CCC(C3CCNC3)CC2)CC1
Cc1cc(C(=O)N2CCC(C3CCNC3)CC2)cc(C)c1OC(F)F
CS(=O)(=O)c1ccccc1C(=O)N1CCC(C2CCNC2)CC1
CCc1ccc(S(C)(=O)=O)cc1C(=O)N1CCC(C2CCNC2)CC1
O=C(c1ccc2[nH]c(C(F)F)nc2c1)N1CCC(C2CCNC2)CC1
O=C(Nc1ccccc1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
O=C(Nc1ccc(Cl)cc1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
Cc1cccc(NC(=O)[C@@H](c2ccccc2)N2Cc3ccccc3C2=O)n1
O=C(Nc1ccncc1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
O=C(Nc1ccc(F)cc1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
COCCNC(=O)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
O=C(NCC1=[SH]C=CC1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
O=C(NCCc1ccccc1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
N#Cc1ccccc1NC(=O)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
O=C(Nc1cccc(F)c1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
O=C(Nc1cccnc1)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O
CNCC1CCCN(C(=O)[C@@H](c2ccccc2)N2Cc3ccccc3C2=O)C1
CN(C)C(=O)C(CNC(=O)[C@@H](c1ccccc1)N1Cc2ccccc2C1=O)c1ccccc1
Design Rationale:
HTS follow up analogs in-stock at Enamine