Submission Details

Molecule(s):
C#Cc1ccc(CNC(=O)N2CCOCC2)cc1

PAT-GYR-359dbb24-1

C#Cc1ccc(CNC(=O)N2CCOCC2)cc1

O=C(NCc1ccc(C#CBr)cc1)N1CCOCC1

PAT-GYR-359dbb24-2

O=C(NCc1ccc(C#CBr)cc1)N1CCOCC1

COC(=O)C#Cc1ccc(CNC(=O)N2CCOCC2)cc1

PAT-GYR-359dbb24-3

COC(=O)C#Cc1ccc(CNC(=O)N2CCOCC2)cc1

NC(=O)C#Cc1ccc(CNC(=O)N2CCOCC2)cc1

PAT-GYR-359dbb24-4

NC(=O)C#Cc1ccc(CNC(=O)N2CCOCC2)cc1

O=C(NCc1ccc(C#CCCO)cc1)N1CCOCC1

PAT-GYR-359dbb24-5

O=C(NCc1ccc(C#CCCO)cc1)N1CCOCC1


Design Rationale:

Expanding fragment x1249

Inspired By:
Discussion: